EP3658552

Aðferð til framleiðslu á N-(5-((4-(4-((dímetýlamínó)metýl)-3-fenýl-1H-pýrasól-1-ýl)pýrimídín-2-ýl)amínó)-4-metoxý-2-morfólínófenýl)akrýlamíði með því að hvarfa tilsvarandi amínið við 3-haló-própíónýl-klóríð

  • Status:
    EP einkaleyfi í gildi á Íslandi
  • EP appl. date:
    25.7.2018
  • EP published:
    13.9.2023
  • EP application number:
    18837360.9
  • Max expiry date:
    24.7.2038
  • Expiry date:
    24.7.2026
  • Next due date:
    31.7.2026
  • Title in English:
    PROCESS FOR PREPARING N-(5-((4-(4-((DIMETHYLAMINO)METHYL)-3-PHENYL-1H-PYRAZOL-1-YL)PYRIMIDIN-2-YL)AMINO)-4-METHOXY-2-MORPHOLINOPHENYL)ACRYLAMIDE BY REACTING THE CORRESPONDING AMINE WITH A 3-HALO-PROPI
  • Language of the patent:
    English

Timeline

Today
25.7.2018EP application
13.9.2023EP Publication
8.11.2023Translation submitted
15.12.2023Registration published
24.7.2026Expires

Owner

  • Name:
    Yuhan Corporation
  • Address:
    74 Noryangjin-ro Dongjak-gu, Seoul 06927, KR

Inventor

  • Name:
    OH, Sang-Ho
  • Address:
    Gunpo-si Gyeonggi-do 15821, KR
  • Name:
    KHOO, Ja-Heouk
  • Address:
    Gunpo-si Gyeonggi-do 15825, KR
  • Name:
    LIM, Jong-Chul
  • Address:
    Yongin-si Gyeonggi-do 17007, KR
  • Name:
    LEE, Seong-Ran
  • Address:
    Suwon-si Gyeonggi-do 16707, KR
  • Name:
    JU, Hyun
  • Address:
    Hwaseong-si Gyeonggi-do 18466, KR
  • Name:
    SHIN, Woo-Seob
  • Address:
    Suwon-si Gyeonggi-do 16697, KR
  • Name:
    PARK, Dae-Gyu
  • Address:
    Suwon-si Gyeonggi-do 16699, KR
  • Name:
    PARK, Su-Min
  • Address:
    Cheongju-si Chungcheongbuk-do 28408, KR
  • Name:
    HWANG, Yoon-Ah
  • Address:
    Suwon-si Gyeonggi-do 16510, KR

Agent

  • Name:
    Árnason Faktor ehf.
  • Address:
    Guðríðarstíg 2-4, 113, Reykjavík,

Priority

  • Number:
    20170096212
  • Date:
    28.7.2017
  • Country:
    KR

Classification

  • Categories:
    C07D 413/14, A61K 31/5377, A61K 31/506

Annual fees

Number

Paid

Expires

Payer

Number: 7

Paid: 6.6.2024

Expires: 24.7.2025

Payer: Árnason Faktor ehf.

Number: 8

Paid: 9.7.2025

Expires: 24.7.2026

Payer: Árnason Faktor ehf.

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